Acetylation of Some Cyclic Enamines With Substituted Acetyl Chlorides
نویسندگان
چکیده
Acylation reaction of a variety of cyclic ketones via acylation of the corresponding enamines is welldefined in the literature. Enamine acylation of carbonyl compounds is a significant synthetic method because of its mildness and the ease of preparing various β-diketones [1-4]. Acylation reactions are performed by means of converting enamines to the enaminoketones and subsequent hydrolysis of the enaminoketones to the desired βdiketones [5,6]. The yield of the reaction is increased when triethylamine is used in the reaction medium as a base to prevent salt formation [7].
منابع مشابه
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